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![[Tyr3]Octreotate](https://aobious.com/aobious/55477/-tyr3-octreotate.jpg "[Tyr3]Octreotate")
View larger Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $74.70 | Total: $7,470.00 |
| 1 | 50 | $86.32 | Total: $4,316.00 |
| 1 | 25 | $101.26 | Total: $2,531.50 |
| 1 | 10 | $119.52 | Total: $1,195.20 |
| 1 | 5 | $141.10 | Total: $705.50 |
Data sheet
| Molecular Formula | C49H64N10O12S2 |
| Molecular Weight | 1049.22 |
| CAS Numbers | 302794-43-0 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(C=1C=2C(NC1)=CC=CC2)[C@H]3NC(=O)[C@H](CC4=CC=C(O)C=C4)NC(=O)[C@@H](NC([C@@H](CC5=CC=CC=C5)N)=O)CSSC[C@@H](C(N[C@@H]([C@@H](C)O)C(O)=O)=O)NC(=O)[C@]([C@@H](C)O)(NC(=O)[C@H](CCCCN)NC3=O)[H] |
| References | Paterson B M, et al. PET imaging of tumours with a 64 Cu labeled macrobicyclic cage amine ligand tethered to Tyr 3-octreotate. Dalton Transactions, 2014, 43[3] 1386-1396. |
More info
[Tyr3]Octreotate is a long peptide compound containing 8 amino acids and is a functional DOTA chelating agent with covalent bonds. [Tyr3]Octreotate binds to transmembrane receptors of SSR2-active NETs and is actively transported into cells by endocytosis, which may increase the required double-stranded DNA breaks and is a potential drug for tumor treatment.