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View larger Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $27.00 | Total: $2,700.00 |
| 1 | 50 | $31.20 | Total: $1,560.00 |
| 1 | 25 | $36.60 | Total: $915.00 |
| 1 | 10 | $43.20 | Total: $432.00 |
| 1 | 5 | $51.00 | Total: $255.00 |
Data sheet
| Molecular Formula | C22H17F4N3O6 |
| Molecular Weight | 495.38 |
| CAS Numbers | 2803881-11-8 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C1N(CC=2C1=CC(COC(NC3=CC(OC(F)(F)F)=CC=C3F)=O)=CC2)C4C(=O)NC(=O)CC4 |
| References | Gerald Gavory, et al. Abstract 3449 Development of MRT-2359, an orally bioavailable GSPT1 molecular glue degrader, for the treatment of lung cancers with MYC-induced translational addiction. Cancer Res. 2023 ; 83[7] 3449. |
More info
MRT-2359 is a potent and orally available GSPT1 reducer with antitumour activity.MRT-2359 inhibits the growth of drug-resistant non-small cell lung cancer (NSCLC) and small cell lung cancer (SCLC) cells.MRT-2359 exhibits preferential activity in MYC-driven cell lines.