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Rare Chemicals
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $48.15 | Total: $4,815.00 |
| 1 | 50 | $55.64 | Total: $2,782.00 |
| 1 | 25 | $65.27 | Total: $1,631.75 |
| 1 | 10 | $77.04 | Total: $770.40 |
| 1 | 5 | $90.95 | Total: $454.75 |
Data sheet
| Molecular Formula | C27H22F2N6O3 |
| Molecular Weight | 516.5 |
| CAS Numbers | 2407854-18-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N#CC1=NC2=C(N(C)C(C([N+]([O-])=O)=C2N3CCN(C(C4=CC=C(C=C4)F)C5=CC=C(C=C5)F)CC3)=O)C=C1 |
| References | Chupak L, et al. Discovery of Potent, Dual-Inhibitors of Diacylglycerol Kinases Alpha and Zeta Guided by Phenotypic Optimization. ACS Med Chem Lett. 2023 Jun 12;14[7] 929-935. |
More info
BMS-502 is a potent dual inhibitor of diacylglycerol kinase (DGK) ? and ? that induces immune responses in human and mouse T cells and blocks intracellular checkpoint signaling in T cells. BMS-502 stimulates immune responses in a dose-dependent manner and can be used to study immune-related diseases.