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NPAS3-IN-1 View larger

NPAS3-IN-1

AT81646

CAS 2207-44-5

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$65.00

$65.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $29.25 Total: $2,925.00
150 $33.80 Total: $1,690.00
125 $39.65 Total: $991.25
110 $46.80 Total: $468.00
15 $55.25 Total: $276.25

Data sheet

Molecular FormulaC10H5N3O2S3
Molecular Weight295.36
CAS Numbers2207-44-5
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeO=[N+]([O-])C1=CN=C(SC2=NC3=C(S2)C=CC=C3)S1
ReferencesLi P, et al. Discovery of a highly potent NPAS3 heterodimer inhibitor by covalently modifying ARNT. Bioorg Chem. 2023 Oct;139 106676.

More info

NPAS3-IN-1 is a potent inhibitor of NPAS3-ARNT heterodimerization, modulating NPAS3 transcription by targeting the interaction between NPAS3 and ARNT at the cellular level.