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Rare Chemicals
- Protein Control Ligand
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $56.70 | Total: $5,670.00 |
| 1 | 50 | $65.52 | Total: $3,276.00 |
| 1 | 25 | $76.86 | Total: $1,921.50 |
| 1 | 10 | $90.72 | Total: $907.20 |
| 1 | 5 | $107.10 | Total: $535.50 |
Data sheet
| Molecular Formula | C15H15N5 |
| Molecular Weight | 265.31 |
| CAS Numbers | 380537-35-9 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN1C=2C(N=C1NN=C(C)C3=CC=CC=N3)=CC=CC2 |
More info
(E)-SI-2 is a potent small-molecule inhibitor of steroid receptor coactivator-3 (SRC-3 or AIB1) that can selectively inhibit the intrinsic transcriptional activities of SRC-3, also inhibits SRC-1 and SRC-2. It selectively reduces cellular protein levels of SRC-3, but not that of CARM-1, blocks MDA-MB-468 cell growth with an IC50 value of 3.4 nM, but spares normal cells.