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View larger Brilanestrant
AT5118
CAS 1365888-06-7
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $34.85 | Total: $174.25 |
| 1 | 10 | $29.52 | Total: $295.20 |
| 1 | 25 | $25.01 | Total: $625.25 |
| 1 | 50 | $21.32 | Total: $1,066.00 |
| 1 | 100 | $18.45 | Total: $1,845.00 |
Data sheet
| Molecular Formula | C26H20ClFN2O2 |
| Molecular Weight | 446.9 |
| CAS Numbers | 1365888-06-7 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCC(=C(c1ccc(C=CC(O)=O)cc1)c1ccc2[nH]ncc2c1)c1ccc(F)cc1Cl |
| References | By Lai, et al. Identification of GDC-0810 [ARN-810], an Orally Bioavailable Selective Estrogen Receptor Degrader [SERD] that Demonstrates Robust Activity in Tamoxifen-Resistant Breast Cancer Xenografts. J Med Chem. 2015 Jun 25;58[12] 4888-904. |
More info
Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM).