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View larger GSK270822A
AT27467
CAS 864082-23-5
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $171.70 | Total: $858.50 |
| 1 | 10 | $145.44 | Total: $1,454.40 |
| 1 | 25 | $123.22 | Total: $3,080.50 |
| 1 | 50 | $105.04 | Total: $5,252.00 |
| 1 | 100 | $90.90 | Total: $9,090.00 |
Data sheet
| Molecular Formula | C24H20N4O2 |
| Molecular Weight | 396.44 |
| CAS Numbers | 864082-23-5 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(NC=1C=C2C(=CC1)NN=C2)(=O)C=3C(CC(=O)NC3C)C4=CC5=C(C=C4)C=CC=C5 |
| References | Identification and Structure-?Function Analysis of Subfamily Selective G Protein-?Coupled Receptor Kinase Inhibitors. By Homan, Kristoff T.; Larimore, Kelly M.; Elkins, Jonathan M.; Szklarz, Marta; Knapp, Stefan; Tesmer, John J. G. From ACS Chemical Biology [2015], 10[1], 310-319. |
More info
GSK270822A is a selective ROCK1 inhibitor. GSK270822A exhibits IC50 of 9nM, 1100nM, 1550nM for ROCK1, RSK1, p70S6K, respectively.