Steroid Hormone Receptors

GSK299115A View larger

GSK299115A

AT27471

CAS 864082-35-9

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$286.00

$286.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $128.70 Total: $12,870.00
150 $148.72 Total: $7,436.00
125 $174.46 Total: $4,361.50
110 $205.92 Total: $2,059.20
15 $243.10 Total: $1,215.50

Data sheet

Molecular FormulaC20H16Cl2N4O2
Molecular Weight415.27
CAS Numbers864082-35-9
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeC(NC=1C=C2C(=CC1)NN=C2)(=O)C=3C(CC(=O)NC3C)C4=CC(Cl)=C(Cl)C=C4
ReferencesGuccione M, et al. G-Protein-Coupled Receptor Kinase 2 [GRK2] Inhibitors Current Trends and Future Perspectives. J Med Chem. 2016 Oct 27;59[20] 9277-9294.

More info

GSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for ROCK1, RSK1, p70S6K, respectively.