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View larger GSK299115A
AT27471
CAS 864082-35-9
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $243.10 | Total: $1,215.50 |
| 1 | 10 | $205.92 | Total: $2,059.20 |
| 1 | 25 | $174.46 | Total: $4,361.50 |
| 1 | 50 | $148.72 | Total: $7,436.00 |
| 1 | 100 | $128.70 | Total: $12,870.00 |
Data sheet
| Molecular Formula | C20H16Cl2N4O2 |
| Molecular Weight | 415.27 |
| CAS Numbers | 864082-35-9 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(NC=1C=C2C(=CC1)NN=C2)(=O)C=3C(CC(=O)NC3C)C4=CC(Cl)=C(Cl)C=C4 |
| References | Guccione M, et al. G-Protein-Coupled Receptor Kinase 2 [GRK2] Inhibitors Current Trends and Future Perspectives. J Med Chem. 2016 Oct 27;59[20] 9277-9294. |
More info
GSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for ROCK1, RSK1, p70S6K, respectively.