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View larger Elacestrant dihydrochloride
AT13675
CAS 1349723-93-8
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $46.80 | Total: $4,680.00 |
| 1 | 50 | $54.08 | Total: $2,704.00 |
| 1 | 25 | $63.44 | Total: $1,586.00 |
| 1 | 10 | $74.88 | Total: $748.80 |
| 1 | 5 | $88.40 | Total: $442.00 |
Data sheet
| Molecular Formula | C30H40Cl2N2O2 |
| Molecular Weight | 531.56 |
| CAS Numbers | 1349723-93-8 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.Cl.CCNCCc1ccc(CN(CC)c2cc(OC)ccc2[C@@H]2CCc3cc(O)ccc3C2)cc1 |
| References | Garner F, et al. RAD1901 a novel, orally bioavailable selective estrogen receptor degrader that demonstrates antitumor activity in breast cancer xenograft models. Anticancer Drugs. 2015 Oct;26[9] 948-56. |
More info
Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ER? and 870 nM for ER?, respectively.