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View larger PROTAC ERR? ligand 1
AT15191
CAS 1264754-13-3
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $11.70 | Total: $1,170.00 |
| 1 | 50 | $13.52 | Total: $676.00 |
| 1 | 25 | $15.86 | Total: $396.50 |
| 1 | 10 | $18.72 | Total: $187.20 |
| 1 | 5 | $22.10 | Total: $110.50 |
Data sheet
| Molecular Formula | C19H11F3N2O4S |
| Molecular Weight | 420.36 |
| CAS Numbers | 1264754-13-3 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O(C1=C(C(F)(F)F)C=C(C#N)C=C1)C2=C(OC)C=C(C=C3C(=O)NC(=O)S3)C=C2 |
| References | Patch RJ, et al. Identification of diaryl ether-based ligands for estrogen-related receptor ? as potential antidiabetic agents. J Med Chem. 2011 Feb 10;54[3] 788-808. |
More info
PROTAC ERR? ligand 1 is an estrogen-related receptor ? (ERR?) antagonist with IC50 values of 0.04 ?M for ERR? and 2.8 ?M for ERR?.