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Steroid Hormone Receptors
- Protein Control Ligand
- Pathway Inhibitors
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- Kinase Inhibitors
- Protease
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- p18
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- p53
- p70
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- Peptidase
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- Ubiquitin-Activating Enzyme
- Adenosine Deaminase
- Clathrin
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- p68
- ACE
- COX
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- Reductase
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- Transferase
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- Transporter Inhibitors
- Cell Inhibition
- Synthase
- Receptor Tyrosine Phosphatases (RTP)
- AChE
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- Autophagy
- Toll-Like Receptor (TLR)
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- G Protein-Coupled Receptor Ligands
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- Angiotensin Receptor
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- CCK Receptors
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- EAA Receptors
- Ghrelin Receptors
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- Histamine Receptors
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- Metabotropic Glutamate Receptors
- Motilin Receptors
- Muscarinic Receptor
- Neuropeptide Receptors
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- Orphan Receptors
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- Purinergic Receptors
- Ryanodine receptor
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- Urotensin Receptor
- Imidazoline receptor
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- β-arrestin/β2-adaptin
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View larger Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $25.65 | Total: $2,565.00 |
| 1 | 50 | $29.64 | Total: $1,482.00 |
| 1 | 25 | $34.77 | Total: $869.25 |
| 1 | 10 | $41.04 | Total: $410.40 |
| 1 | 5 | $48.45 | Total: $242.25 |
Data sheet
| Molecular Formula | C10H13ClN4O2 |
| Molecular Weight | 256.69 |
| CAS Numbers | 862892-90-8 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCCCCn1c2nc(Cl)[nH]c2c(=O)[nH]c1=O |
| References | Dobbins RL, et al. GSK256073, a selective agonist of G-protein coupled receptor 109A [GPR109A] reduces serum glucose in subjects with type 2 diabetes mellitus.Diabetes Obes Metab. |
More info
GSK256073 is an orally active GPR109A agonist. GSK256073 also is a long-lasting and non-flushing HCA2 (hydroxy-carboxylic acid receptor 2) full agonist (pEC50: 7.5). GSK256073 acutely improves glucose homeostasis via inhibition of lipolysis.