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Steroid Hormone Receptors
- Protein Control Ligand
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $16.20 | Total: $1,620.00 |
| 1 | 50 | $18.72 | Total: $936.00 |
| 1 | 25 | $21.96 | Total: $549.00 |
| 1 | 10 | $25.92 | Total: $259.20 |
| 1 | 5 | $30.60 | Total: $153.00 |
Data sheet
| Molecular Formula | C8H8N2O2 |
| Molecular Weight | 164.16 |
| CAS Numbers | 1268882-43-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | [H][C@]12C[C@@]1([H])c1[nH]nc(C(O)=O)c1C2 |
| References | Boatman PD, et al. [1aR,5aR]1a,3,5,5a-Tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid [MK-1903] a potent GPR109a agonist that lowers free fatty acids in humans. J Med Chem. 2012;55[8] 3644-3666. |
More info
MK 1903 is a potent and selective complete agonist for the hydroxy-carboxylic acid receptor 2 (HCA2). HCA2 is also known as G protein-coupled receptor 109A(GPR109A). MK 1903 reduced Foschlin-induced cAMP production in uniform time-resolved fluorescence (htf) measurements using CHO cells expressing the human receptor (ECso-12.9 nM).