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View larger PROTAC ERR? ligand 2
AT5835
CAS 2306388-57-6
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $43.35 | Total: $216.75 |
| 1 | 10 | $36.72 | Total: $367.20 |
| 1 | 25 | $31.11 | Total: $777.75 |
| 1 | 50 | $26.52 | Total: $1,326.00 |
| 1 | 100 | $22.95 | Total: $2,295.00 |
Data sheet
| Molecular Formula | C20H13F6NO4 |
| Molecular Weight | 445.31 |
| CAS Numbers | 2306388-57-6 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1cc(C=C(C#N)C(O)=O)ccc1OCc1ccc(cc1C(F)(F)F)C(F)(F)F |
| References | Peng L , Zhang Z , Lei C , et al. Identification of New Small-Molecule Inducers of Estrogen-Related Receptor alpha [ERRa] Degradation[J]. ACS Medicinal Chemistry Letters, 2019, 10[5]. |
More info
PROTAC ERR? ligand 2 is an inverse agonist for the estrogen-related receptor ? (ERR?) with an IC50 of 5.67 nM.