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View larger Icenticaftor
AT9499
CAS 1334546-77-8
1000 Items
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $196.35 | Total: $981.75 |
| 1 | 10 | $166.32 | Total: $1,663.20 |
| 1 | 25 | $140.91 | Total: $3,522.75 |
| 1 | 50 | $120.12 | Total: $6,006.00 |
| 1 | 100 | $103.95 | Total: $10,395.00 |
Data sheet
| Molecular Formula | C12H13F6N3O3 |
| Molecular Weight | 361.24 |
| CAS Numbers | 1334546-77-8 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1nc(C(=O)NC[C@](C)(O)C(F)(F)F)c(N)cc1C(F)(F)F |
| References | Darren Le Grand, et al. Discovery of Icenticaftor [QBW251], a Cystic Fibrosis Transmembrane Conductance Regulator Potentiator with Clinical Efficacy in Cystic Fibrosis and Chronic Obstructive Pulmonary Disease. J Med Chem. 2021 Jun 10;64[11] 7241-7260. |
More info
Icenticaftor (QBW251) is an orally active potentiator of the CFTR channel.