Ubiquitin-Activating Enzyme

IMP-1710 View larger

IMP-1710

AT37591

CAS 2383117-96-0

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$253.00

$253.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $113.85 Total: $11,385.00
150 $131.56 Total: $6,578.00
125 $154.33 Total: $3,858.25
110 $182.16 Total: $1,821.60
15 $215.05 Total: $1,075.25

Data sheet

Molecular FormulaC23H19N5O
Molecular Weight381.43
CAS Numbers2383117-96-0
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeC(=O)(N1C=2C(=C(C=CC2)C=3C=4C(NC3)=NC=C(C#C)C4)CC1)[C@H]5N(C#N)CCC5
ReferencesPanyain, N., Godinat, A., Lanyon-Hogg, T., et al.Discovery of a potent and selective covalent inhibitor and activity-based probe for the deubiquitylating enzyme UCHL1, with antifibrotic activityJ. Am. Chem. Soc.142[28]12020-12026[2020]

More info

IMP-1710 is a selective UCH-L1 inhibitor with an IC50 value of 38 nM in a fluorescence polarization assay.