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View larger TRPV4 agonist-1 free base
AT13214L
CAS 2314467-59-7
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $21.60 | Total: $2,160.00 |
| 1 | 50 | $24.96 | Total: $1,248.00 |
| 1 | 25 | $29.28 | Total: $732.00 |
| 1 | 10 | $34.56 | Total: $345.60 |
| 1 | 5 | $40.80 | Total: $204.00 |
Data sheet
| Molecular Formula | C25H22F2N4O2 |
| Molecular Weight | 448.46 |
| CAS Numbers | 2314467-59-7 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN1CCN(CC1)c1nc2c(F)cccc2c(=O)n1-c1ccc(Oc2ccc(F)cc2)cc1 |
| References | Atobe M, et al. Discovery of Novel Transient Receptor Potential Vanilloid 4 [TRPV4] Agonists as Regulators of Chondrogenic Differentiation Identification of Quinazolin-4[3 H]-ones and in Vivo Studies on a Surgically Induced Rat Model of Osteoarthritis. J Med Chem. 2019 Jan 28. |
More info
TRPV4 agonist-1 free base (OUN67600) is an agonist of transient receptor potential vanilloid 4 (TRPV4;EC50 of 60 nM, in the hTRPV4 Ca2+ assay).