Votage-Gated Ion Channel Blockers

OMDM-5 View larger

OMDM-5

AT12306

CAS 616884-66-3

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$126.00

$126.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $56.70 Total: $5,670.00
150 $65.52 Total: $3,276.00
125 $76.86 Total: $1,921.50
110 $90.72 Total: $907.20
15 $107.10 Total: $535.50

Data sheet

Molecular FormulaC26H44N2O3
Molecular Weight432.64
CAS Numbers616884-66-3
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeC(NNC(CCCCCCCC=CCCCCCCCC)=O)C1=CC(OC)=C(O)C=C1
ReferencesOrtar G, et al. Novel selective and metabolically stable inhibitors of anandamide cellular uptake. Biochem Pharmacol. 2003 May 1;65[9] 1473-81.

More info

OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 ?M). OMDM-5 is a selective anandamide cellular uptake (ACU) inhibitor(Ki = 4.8 ?M).