Votage-Gated Ion Channel Blockers

TC-N 1752 View larger

TC-N 1752

AT23439

CAS 1211866-85-1

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$43.00

$43.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $19.35 Total: $1,935.00
150 $22.36 Total: $1,118.00
125 $26.23 Total: $655.75
110 $30.96 Total: $309.60
15 $36.55 Total: $182.75

Data sheet

Molecular FormulaC25H27F3N6O3
Molecular Weight516.52
CAS Numbers1211866-85-1
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(OC(F)(F)F)cc2)c1C
ReferencesLin Z, et, al. Biophysical and Pharmacological Characterization of Nav1.9 Voltage Dependent Sodium Channels Stably Expressed in HEK-293 Cells. PLoS One. 2016 Aug 24;11[8] e0161450.

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TC-N 1752 is an orally active inhibitor of Nav1.7 channel with IC50 of 0.17 ?M. TC-N 1752 shows analgesic activities.