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View larger (S)-ABT 102
AT29522L
CAS 808756-70-9
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $84.15 | Total: $420.75 |
| 1 | 10 | $71.28 | Total: $712.80 |
| 1 | 25 | $60.39 | Total: $1,509.75 |
| 1 | 50 | $51.48 | Total: $2,574.00 |
| 1 | 100 | $44.55 | Total: $4,455.00 |
Data sheet
| Molecular Formula | C21H24N4O |
| Molecular Weight | 348.44 |
| CAS Numbers | 808756-70-9 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(C(NC1=C2C(NN=C2)=CC=C1)=O)[C@@H]3C=4C(=CC(C(C)(C)C)=CC4)CC3 |
| References | Gomtsyan A, et al. Identification of [R]-1-[5-tert-butyl-2,3-dihydro-1H-inden-1-yl]-3-[1H-indazol-4-yl]urea [ABT-102] as a potent TRPV1 antagonist for pain management. J Med Chem. 2008 Feb 14;51[3] 392-5. |
More info
N-[(1S)-5-tert-butyl-2,3-dihydro-1H-inden-1-yl]-N'-1H-indazol-4-ylurea is a potent TRPV1 antagonist, blocking activation of TRPV1 by capsaicin with the IC50 of 123 nM.