Votage-Gated Ion Channel Blockers

Obafistat View larger

Obafistat

AT39635

CAS 2160582-57-8

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$57.00

$57.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $25.65 Total: $2,565.00
150 $29.64 Total: $1,482.00
125 $34.77 Total: $869.25
110 $41.04 Total: $410.40
15 $48.45 Total: $242.25

Data sheet

Molecular FormulaC15H16FN5O3S
Molecular Weight365.38
CAS Numbers2160582-57-8
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeFc1cccc(c1)S(=O)(=O)N1C2CCC1CN(C2)C(=O)c1cnn[nH]1
ReferencesMarcus Koppitz, et al. [8-[phenylsulfonyl]-3,8-diazabicyclo[3.2.1]oct-3-yl] [1h-1,2,3-triazol-4-yl]methanones. WO2017202817A1.

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Obafistat is a potent inhibitor of aldo-keto reductase AKR1C3 with an IC50 of 1.2 nM for human AKR1C3.