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GSK5182
AOB1629
CAS No: 877387-37-6
AOBIOUS launched this product in 2015
CITATIONS - Publications That Use AOBIOUS Product
1) Nat Commun. 2018; 9: 1920 and JUSTIA Patent 2018
2) Biochemical and Biophysical Res Commun V563, P15(2021)
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $16.88 | Total: $1,687.50 |
| 1 | 50 | $19.50 | Total: $975.00 |
| 1 | 25 | $22.88 | Total: $571.88 |
| 1 | 10 | $27.00 | Total: $270.00 |
| 1 | 5 | $31.88 | Total: $159.38 |
Data sheet
| Molecular Formula | C27H31NO3 |
| Molecular Weight | 417.54 |
| CAS Numbers | 877387-37-6 |
| Storage Condition | 0°C (short term), -20°C (long term), desiccated |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| Synonym | GSK5182; GSK 5182; GSK-5182. |
| IUPAC/Chemical Name | 4-[(Z)-1-[4-(2-dimethylaminoethoxy)phenyl]-5-hydroxy-2-phenylpent-1-enyl]phenol |
| InChl Key | ZVSFNBNLNLXEFQ-RQZHXJHFSA-N |
| InChl Code | InChI=1S/C27H31NO3/c1-28(2)18-20-31-25-16-12-23(13-17-25)27(22-10-14-24(30)15-11-22)26(9-6-19-29)21-7-4-3-5-8-21/h3-5,7-8,10-17,29-30H,6,9,18-20H2,1-2H3/b27-26- |
| SMILES Code | OC1=CC=C(/C(C2=CC=C(OCCN(C)C)C=C2)=C(C3=CC=CC=C3)CCCO)C=C1 |
| References | 1) Joo J, Wu Z, Lee B, Shon JC, Lee T, Lee IK, Sim T, Kim KH, Kim ND, Kim SH, Liu KH. In vitro metabolism of an estrogen-related receptor γ modulator, GSK5182, by human liver microsomes and recombinant cytochrome P450s. Biopharm Drug Dispos. 2015 Apr;36(3):163-73. doi: 10.1002/bdd.1929. PubMed PMID: 25451157. |
More info
Novel inverse agonist of estrogen-related receptor γ (ERRγ)
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