Enzyme Inhibitors

LEI110 View larger

LEI110

AOB17659

CAS: 2313525-90-3

 

Chemical Name: KB-2115; 3-[3,5-Dibromo-4-(4-hydroxy-3-propan-2-ylphenoxy)anilino]-3-oxopropanoic acid

More details

Molarity Calculation Cart®

HOW TO ORDER

$37.00

$37.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $16.65 Total: $1,665.00
150 $19.24 Total: $962.00
125 $22.57 Total: $564.25
110 $26.64 Total: $266.40
15 $31.45 Total: $157.25

Data sheet

Molecular FormulaC25H23F3N2O3
Molecular Weight456.47
CAS Numbers2313525-90-3
Storage Condition0°C (short term), -20°C (long term), desiccated
SolubilityDMSO
Purity98% by HPLC
SynonymLEI 110; LEI-110
IUPAC/Chemical Name2-oxo-5-phenyl-N-(4-((5-(trifluoromethyl)pyridin-2-yl)oxy)phenethyl)pentanamide
References1) Zhou J, et al. ACS Chem Biol. 2019 Jan 8. doi: 10.1021/acschembio.8b00969.

More info

Novel potent PLA2G16 inhibitor (Ki = 20 nM), selectively pan-inhibiting the HRASLS family of thiol hydrolases (i.e., PLA2G16, HRASLS2, RARRES3 and iNAT), reducing cellular arachidonic acid levels and oleic acid-induced lipolysis in human HepG2 cells

Customers who bought this product also bought: